1-(9,10-Dihydro-6H-6,10-methanoazepino[4,5-g]-quinoxalin-8(7H)-yl)-2,2,2-trifluoroethanone

Synonym
Product Category
Product Code
CAS Number
MDL Number
Pubchem SID
Reaxys RN

Trifluoromethyl Building Blocks
KUMI3F173
230615-70-0
 
11483621

image-155171-Trimethyl(trifluoromethyl)silane_reagent.png
Chemical Name
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1-(9,10-Dihydro-6H-6,10-methanoazepino[4,5-g]-quinoxalin-8(7H)-yl)-2,2,2-trifluoroethanone
C15H12F3N3O
307.27
≥98%
White to Yellow Solid
162-164°C
5g,10g,25g,50g,100g,250g and 500g
Store at room temperature
1-(9,10-Dihydro-6H-6,10-methanoazepino[4,5-g]-quinoxalin-8(7H)-yl)-2,2,2-trifluoroethanone is a trifluoromethylated pharmaceutical intermediate typically used as protected impurity to prepare varenicline for smoking cessation.
Varenicline: an alpha4beta2 nicotinic receptor partial agonist for smoking cessation. [1]
Reference:
[1] J.W.Coe, et al, J. Med. Chem., 2005, 48(10), pp 3474-3477.
Signal Word
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HS Code
RIDADR
Legal Information
Not classified as a hazardous substance or mixture


2933990090
NONH for all modes of transport

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