2-Amino-9-[(1S,3R,4S)-4-hydroxy-3-(hydroxymethyl)-2-methylidenecyclopentyl]-3H-purin-6-one

Synonym
Product Category
Product Code
CAS Number
MDL Number
Pubchem CID
Reaxys RN
Entecavir,  Baraclude
API & Intermediates
KAPI0F37
142217-69-4
MFCD11046562 
153941
7692760
image-155171-Trimethyl(trifluoromethyl)silane_reagent.png
Chemical Name
Molecular Formula
Molecular Weight
Assay
Appearance
Melting Point
Packaging
Storage
2-Amino-9-[(1S,3R,4S)-4-hydroxy-3-(hydroxymethyl)-2-methylidenecyclopentyl]-3H-purin-6-one
C12H15O3N5
277.28
≥98% (HPLC)
White to Off-white Solid
249-252°C
5g,10g,25g,50g,100g,250g and 500g
Store at 2-8°C temp.
Entecavir is an antiviral guanine analog that inhibits reverse transcription, DNA replication and transcription in the viral replication process. It is typically used to treat hepatitis B virus infection.
Identification of BMS-200475 as a potent and selective inhibitor of hepatitis B virus. [1]
Entecavir: a potent new antiviral drug for hepatitis B. [2]
A comparison of entecavir and lamivudine for HBeAg-positive chronic hepatitis B. [3]
References:
[1] S.F.Innaimo, et al, Antimicrob. Agents Chemother., 1997, 41(7), pp 1444-1448.
[2] P.Honkoop, et al, Expert Opin. Investig. Drugs, 2003, 12(4), pp 683-688.
[3] T.T.Chang, et al, N. Engl. J. Med., 2006, 354(10), pp 1001-1010.
Signal Word
Hazard Statements
Precautionary Statements
HS Code
RIDADR
RETCS
Legal Information
Not classified as a hazardous substance or mixture


2933599590
NONH for all modes of transport


1. Product Specification
2. Safety Data Sheet
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