2-Bromo-5-(bromomethyl)pyridine

Synonym
Product Category
Product Code
CAS Number
MDL Number
Pubchem CID
Reaxys RN
2-Bromo-5-pyridylmethyl bromide
API & Intermediates
KUMI0F953
101990-45-8
MFCD11656267
6424660
1635694
image-155171-Trimethyl(trifluoromethyl)silane_reagent.png
Chemical Name
Molecular Formula
Molecular Weight
Assay
Appearance
Melting Point
Packaging
Storage
2-Bromo-5-(bromomethyl)pyridine
C6H5Br2N
250.92
≥98%
White to Brown Solid
60-65°C
5g,10g,20g,50g,100g,500g and 1kg
Store at 2-8°C temp.
 2-Bromo-5-(bromomethyl)pyridine is a pharmaceutical intermediate typically used for the preparation of positive allosteric modulators (PAMs) of the M1 receptor, SRC kinase inhibitors and selective CYP11B1 inhibitors.
4-Anilino-7-pyridyl-3-quinolinecarbonitriles as Src kinase inhibitors. [1]
First selective CYP11B1 inhibitors for the treatment of cortisol-dependent diseases. [2]
Selective allosteric modulation of muscarinic acetylcholine receptors for the treatment of schizophrenia and substance use disorders. [3]
References:
[1] N.Zhang, et al, Bioorg. Med. Chem., 2009, 19(17), pp 5071-5074.
[2] U.E.Hille, et al, ACS Med. Chem. Lett., Bioorg. Med. Chem., 2009, 19(17), pp 5071-5074.
[3] L.B.Teal, et al, Adv. Pharmacol., 2019, 86, pp 153-196.
Signal Word
Hazard Statements
Precautionary Statements
HS Code
RIDADR
Legal Information
Warning
H302,H315,H319,H335
P261,P305+P351+P338
2933399990
NONH for all modes of transport

1. Product Specification
2. Safety Data Sheet
Please inquire for pricing and availability of this product by writing email to sales@kumidas.com.