(3S,4S)-tert-butyl 3-amino-4-fluoropyrrolidine-1-carboxylate

Synonym
Product Category
Product Code
CAS Number
MDL Number
Pubchem CID
Reaxys RN
Trans-1-Boc-3-amino-4-fluoropyrrolidine
Fluorinated Building Blocks
KUMI1F58
1363382-79-9
MFCD18207795
45489881
19510565
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Chemical Name
Molecular Formula
Molecular Weight
Assay
Appearance
Melting Point
Packaging
Storage
(3S,4S)-tert-butyl 3-amino-4-fluoropyrrolidine-1-carboxylate
C9H17FN2O2
204.24
≥97%
Solid

1g,5g,10g,25g and 50g
Store at room temperature
(3S,4S)-tert-butyl 3-amino-4-fluoropyrrolidine-1-carboxylate (trans-1-Boc-3-amino-4-fluoropyrrolidine) is a useful fluorinated building block in the synthesis of various pharmaceutically and biologically active compounds, e.g. preparation of aminopyrrolidine factor Xa inhibitors (as anticogulants), bruton's tyrosine kinase and selectively substituted quinoline compounds that act as antagonists or inhibitors for Toll-like receptors 7 and/or 8.
Design of novel aminopyrrolidine factor Xa inhibitors from a screening hit. [1]
Reference:
[1] K.G.Zbinden, et al, Eur. J. Med. Chem., 2009, 44(7), pp 2787-2795.
Signal Word
Hazard Statements
Precautionary Statements
HS Code
RIDADR
Legal Information
Warning
H302,H335
P261,P280,P305+P351+P338

NONH for all modes of transport

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